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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T36848 | Combretastatin A-1 | Combretastatin A1 | Akt , Microtubule Associated |
Combretastatin A-1 is a potent microtubule inhibitor with anti-tumour and anti-vascular activity, acting through microtubule protein depolymerisation-mediated inactivation of AKT to inhibit the Wnt/β-catenin pathway, and... | |||
T12404 | CCK-A receptor inhibitor 1 | cholecystokinin | |
CCK-A receptor inhibitor 1 is a potent inhibitor of the cholecystokinin A (CCK-A) receptor (IC50: 340 nM).CCK-A receptor inhibitor 1 can be used for the study of diseases related to the digestive system. | |||
TP1179L | Porcine dynorphin A(1-13) acetate | Dynorphin A Porcine Fragment 1-13 acetate,Porcine dynorphin A(1-13) acetate(72957-38-1 free base) | Opioid Receptor |
Porcine dynorphin A(1-13) acetate (Dynorphin A Porcine Fragment 1-13 acetate) is a potent, endogenous κ opioid receptor agonist and is antinociceptive at physiological concentrations. Exposure to dynorphin A (1-13) cause... | |||
T76341L | [DPro10] Dynorphin A (1-11)acetate,porcine | [DPro10] Dynorphin A (1-11)acetate,porcine(94596-26-6 Free base) | Opioid Receptor |
[DPro10] Dynorphin A (1-11)acetate,porcine is a highly potent κ-opioid receptor agonist with a Ki value of 0.13 nM. [DPro10] Dynorphin A (1-11), porcine is an n-alkylated derivative with analgesic activity. | |||
TP1813L | Dynorphin A 1-10 acetate(79994-24-4 free base) | Opioid Receptor | |
Dynorphin A (1-10) acetate is an endogenous opioid neuropeptide, binds to extracellular loop 2 of the κ-opioid receptor. Dynorphin A (1-10) also blocks NMDA-activated current with an IC50 of 42.0 μM. | |||
T21708L | Angiotensin 1/2 + A (2 - 8) Acetate | Angiotensin 1/2 + A (2 - 8) Acetate (51833-76-2 Free base) | Others |
Angiotensin 1/2 + A (2 - 8) Acetate is a Vasoconstrictor. | |||
T4924 | α-D-Glucose-1-phosphate disodium | α-D-Glucose 1-phosphate disodium salt hy,α-D-Glucopyranose 1-phosphate | Others , Endogenous Metabolite |
α-D-Glucose 1-phosphate disodium salt is converted into D-glucose-6-phosphate by the enzyme phosphoglucomutase. | |||
T38817 | Golgicide A-1 | GCA-1,Golgicide A-1 | |
Golgicide A-1 (GCA-1) is a moderately potent cis-diastereomer variant of Golgicide A (GCA) specifically designed to inhibit mosquito reproduction. | |||
T21781 | A-286982 | Integrin | |
A 286982 is an inhibitor that blocks the integrin-ligand interaction between leukocyte function-associated antigen-1 (LFA-1) and intercellular adhesion molecule-1. | |||
T11373 | GCN2-IN-1 | A-92 | Others |
GCN2-IN-1 (A-92) is an effective GCN2 inhibitor and can be used in research on the treatment of cancer as a chemotherapeutic agent. | |||
T10927 | Cyt-PTPε Inhibitor-1 | Cyt-PTP|A Inhibitor-1 | Phosphatase , Src |
Cyt-PTPε Inhibitor-1 (A Inhibitor-1) is an inhibitor of cytosolic protein tyrosine phosphatase ε. Cyt-PTPε Inhibitor-1 blocks the dephosphorylation of c-Src and exhibits anti-osteoclastic activity. | |||
TN1517 | 1-(2,6-dimethoxyphenyl)-3-(4-hydroxyphenyl)propan-1-one | Cochinchinenin A | Others |
1-(2,6-dimethoxyphenyl)-3-(4-hydroxyphenyl)propan-1-one (Cochinchinenin A) is the material basis for the analgesic effect of Dragons Blood. | |||
T39778 | Influenza A virus-IN-1 | ||
Influenza A virus-IN-1, a dihydropyrrolidones derivative, is a highly effective inhibitor of various subtypes of influenza A virus (IAV) with IC 50 values ranging from 3.11 μM to 7.13 μM. It effectively suppresses IAV re... | |||
T36432 | A2ti-1 | Virus Protease | |
A2ti-1 is a highly selective inhibitor of annexin A2/S100A10 heterotetramer (A2t) (IC50: 24 μM) that inhibits ARV-mediated activation of Src and p38 mitogen-activated protein kinase (MAPK). A2ti-1 can be used to study hu... | |||
T2254 | A-205804 | Integrin | |
A-205804 is a specific and effective inhibitor of E-selectin( IC50=20 nM ) and ICAM-1(IC50=25 nM) expression. | |||
T40367 | Combretastatin A-1 phosphate tetrasodium | Combretastatin A-1 phosphate tetrasodium,OXi-4503 tetrasodium | |
Combretastatin A-1 phosphate (OXi-4503) tetrasodium, a prodrug of Combretastatin A-1, is a tubulin-binding microtubule polymerization inhibitor that targets the colchicine-binding site. By inducing tubulin depolymerizati... | |||
TN2525 | 1-Acetyltagitinin A | Others | |
1-Acetyltagitinin A is a natural product of Tithonia, Asteraceae. The catalog number is TN2525 and the CAS number is 60547-63-9. 1-Acetyltagitinin A can be used as a reference standard. | |||
T30222 | Avenacin A 1 | ||
Avenacin A 1 is a biochemical. | |||
T29787 | Ajugamarin A 1 | ||
Ajugamarin A 1 is a Neoclerodane diterpenoid. | |||
TP1813 | Dynorphin A (1-10) | Dynorphin A 1-10 | |
Dynorphin A (1-10), an endogenous opioid neuropeptide, interacts with the κ-opioid receptor by binding to its extracellular loop 2 and inhibits NMDA-activated current, demonstrating an IC50 value of 42.0 μM. |